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WEB 2086, Tocris Bioscience™

Catalog No. 233910
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Quantity:
1 mg
10 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Potent PAF receptor antagonist

Potent, selective platelet-activating factor (PAF) receptor antagonist (Ki = 16.3 nM). Displays anti-inflammatory, antiangiogenic and anticancer activity. Inhibits growth and proliferation of MCF-7 breast cancer cells.

Chemical Identifiers

CAS 105219-56-5
Molecular Formula C22H22ClN5O2S
Molecular Weight (g/mol) 455.961
InChI Key JGPJQFOROWSRRS-UHFFFAOYSA-N
Synonym apafant, apafanto, apafantum, triazolodiazepine, apafant usan:inn, apafantum inn-latin, apafanto inn-spanish, web 2086bs, unii-j613ni05sv, 3h apafant
PubChem CID 65889
SMILES CC1=NN=C2N1C3=C(C=C(S3)CCC(=O)N4CCOCC4)C(=NC2)C5=CC=CC=C5Cl

Specifications

Quantity 10 mg
Formula Weight 455.96
Percent Purity >99%
Chemical Name or Material WEB 2086

Safety and Handling

Recommended Storage Desiccate at +4°C
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