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  7. VU 10010, Tocris Bioscience™

VU 10010, Tocris Bioscience™

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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
633283-39-3
C17H16ClN3OS
345.845
FPRULFHDSFKYBV-UHFFFAOYSA-N
3-amino-n-4-chlorophenyl methyl-4,6-dimethylthieno 2,3-b pyridine-2-carboxamide, 3-amino-n-4-chlorobenzyl-4,6-dimethylthieno 2,3-b pyridine-2-carboxamide, 2fli, 2-fly, f-ligrlo-nh2, 2-fap, 2-f-ligrlo-nh2, d0n2vn, 2-furoyl-ligrlo-amide trifluoroacetate salt, 2-furoyl-leu-ile-gly-arg-leu-orn-nh2 trifluoroacetate salt
714286
3-amino-N-[(4-chlorophenyl)methyl]-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide
CC1=CC(=NC2=C1C(=C(S2)C(=O)NCC3=CC=C(C=C3)Cl)N)C
This item is not returnable. View return policy
633283-39-3
C17H16ClN3OS
345.845
FPRULFHDSFKYBV-UHFFFAOYSA-N
3-amino-n-4-chlorophenyl methyl-4,6-dimethylthieno 2,3-b pyridine-2-carboxamide, 3-amino-n-4-chlorobenzyl-4,6-dimethylthieno 2,3-b pyridine-2-carboxamide, 2fli, 2-fly, f-ligrlo-nh2, 2-fap, 2-f-ligrlo-nh2, d0n2vn, 2-furoyl-ligrlo-amide trifluoroacetate salt, 2-furoyl-leu-ile-gly-arg-leu-orn-nh2 trifluoroacetate salt
714286
3-amino-N-[(4-chlorophenyl)methyl]-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide
CC1=CC(=NC2=C1C(=C(S2)C(=O)NCC3=CC=C(C=C3)Cl)N)C

Description

Selective allosteric potentiator of M4 receptors

Selective allosteric potentiator of M4 acetylcholine receptors (EC50 values are 33 and 0.7 nM for ACh in the absence and presence of VU10010 respectively). Binds to an allosteric site on the receptor increasing affinity for ACh and coupling to G-proteins.
Quantity 50 mg
Formula Weight 345.85
Percent Purity >99%
Chemical Name or Material VU 10010

Safety and Handling

Recommended Storage : Store at +4°C