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OPC 21268, Tocris Bioscience™

Catalog No. 392450
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Quantity:
10 mg
50 mg
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This item is not returnable. View return policy

Description

Orally active vasopressin V1 antagonist

Nonpeptide vasopressin V1 receptor antagonist. Displays greater affinity for rat V1 than human V1 (Ki values are 25 and 8800 nM respectively). Exhibits 1000-fold selectivity for V1 receptors over V2 receptors. Orally active.

Chemical Identifiers

CAS 131631-89-5
Molecular Formula C26H31N3O4
Molecular Weight (g/mol) 449.551
InChI Key KSNUCNRMDYJBKT-UHFFFAOYSA-N
Synonym fuscoside, 1-1-4-3-acetylaminopropoxy benzoyl-4-piperidyl-3,4-dihydro-2 1h-quinolinone, opc-21268 hydrate, n-3-4-4-2-oxo-3,4-dihydroquinolin-1-yl piperidine-1-carbonyl phenoxy propyl acetamide, acetamide, n-3-4-4-3,4-dihydro-2-oxo-1 2h-quinolinyl-1-piperidinyl carbonyl phenoxy propyl, n-3-4-4-2-oxo-3,4-dihydroquinolin-1 2h-yl piperidine-1-carbonyl phenoxy propyl acetamide, acmc-20mu6h, d03qhk, d08oro, n-3-4-4-2-oxo-3,4-dihydro-2h-quinolin-1-yl-piperidine-1-carbonyl-phenoxy-propyl-acetamide
PubChem CID 114904
IUPAC Name N-[3-[4-[4-(2-oxo-3,4-dihydroquinolin-1-yl)piperidine-1-carbonyl]phenoxy]propyl]acetamide
SMILES CC(=O)NCCCOC1=CC=C(C=C1)C(=O)N2CCC(CC2)N3C(=O)CCC4=CC=CC=C43

Specifications

Quantity 50 mg
Formula Weight 449.54
Percent Purity >98%
Chemical Name or Material OPC 21268

Safety and Handling

Recommended Storage Store at +4°C
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