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Gavestinel, Tocris Bioscience™

Catalog Number 234850
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
153436-38-5
C18H12Cl2N2NaO3
398.195
OBPMZHMRJJJUBC-UHDJGPCESA-N
gavestinel
67241466
3-[(E)-3-anilino-3-oxoprop-1-enyl]-4,6-dichloro-1H-indole-2-carboxylic acid;sodium
C1=CC=C(C=C1)NC(=O)C=CC2=C(NC3=CC(=CC(=C32)Cl)Cl)C(=O)O.[Na]
This item is not returnable. View return policy
153436-38-5
C18H12Cl2N2NaO3
398.195
OBPMZHMRJJJUBC-UHDJGPCESA-N
gavestinel
67241466
3-[(E)-3-anilino-3-oxoprop-1-enyl]-4,6-dichloro-1H-indole-2-carboxylic acid;sodium
C1=CC=C(C=C1)NC(=O)C=CC2=C(NC3=CC(=CC(=C32)Cl)Cl)C(=O)O.[Na]

Description

Potent and selective glycine site antagonist; orally available and active in vivo

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites. Orally bioavailable and active in vivo.
Quantity 50 mg
Formula Weight 397.19
Percent Purity >98%
Chemical Name or Material Gavestinel

Safety and Handling

Recommended Storage Desiccate at Room Temperature
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