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JZP 361, >99%, Tocris Bioscience™
Potent and selective reversible MAGL inhibitor
Supplier: R&D Systems 5851/50
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Description
Potent and selective reversible MAGL inhibitor (IC50 = 46 nM). Exhibits 35-fold and 150-fold higher selectivity over human FAAH and ABHD6, respectively (IC50 values are 1.79 and 7.24 μM, respectively). Displays affinity for H1 receptors (pA2 = 6.81). Exhibits no activity at cannabinoid receptors at 10 μM.Specifications
[4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl](1H-1,2,4- | |
>99% | |
50 mg | |
405.88 |
1680193-80-9 | |
C22H20ClN5O | |
Soluble to 100mM in DMSO and to 20mM in ethanol |
Safety and Handling
Recommended Storage : Store at 4deg;C
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