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T 98475, Tocris Bioscience™

Catalog Number 25191
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Quantity:
1 mg
This item is not returnable. View return policy
199119-18-1
C37H37F2N3O4S
657.777
RANJJVIMTOIWIN-UHFFFAOYSA-N
unii-f1klt23o3a, f1klt23o3a, chembl71917, 7-2,6-difluorophenyl methyl-4,7-dihydro-2-4-2-methyl-1-oxopropyl amino phenyl-3-methyl phenylmethyl amino methyl-4-oxo-thieno 2,3-b pyridine-5-carboxylic acid 1-methylethyl ester, d02nco, isopropyl 3-benzyl methyl amino methyl-7-2,6-difluorophenyl methyl-2-4-2-methylpropanoylamino phenyl-4-oxo-thieno 2,3-b pyridine-5-carboxylate, isopropyl 3-n-benzyl-n-methylaminomethyl-7-2,6-difluorobenzyl-4,7-dihydro-2-4-isobutyrylaminophenyl-4-oxothieno 2,3-b pyridine-5-carboxylate hydrochloride, propan-2-yl 3-benzyl methyl amino methyl-7-2,6-difluorophenyl methyl-2-4-2-methylpropanoylamino phenyl-4-oxothieno 2,3-b pyridine-5-carboxylate, thieno 2,3-b pyridine-5-carboxylic acid, 7-2,6-difluorophenyl methyl-4,7-dihydro-2-4-2-methyl-1-oxopropyl amino phenyl-3-methyl phenylmethyl amino methyl-4-oxo-, 1-methylethyl ester, hydrochloride, 3-benzyl-methyl-amino-methyl-7-2,6-difluoro-benzyl-2-4-isobutyrylamino-phenyl-4-oxo-4,7-dihydro-thieno 2,3-b pyridine-5-carboxylic acid isopropyl ester; hydrochloride
9874838
propan-2-yl 3-[[benzyl(methyl)amino]methyl]-7-[(2,6-difluorophenyl)methyl]-2-[4-(2-methylpropanoylamino)phenyl]-4-oxothieno[2,3-b]pyridine-5-carboxylate
CC(C)C(=O)NC1=CC=C(C=C1)C2=C(C3=C(S2)N(C=C(C3=O)C(=O)OC(C)C)CC4=C(C=CC=C4F)F)CN(C)CC5=CC=CC=C5
This item is not returnable. View return policy
199119-18-1
C37H37F2N3O4S
657.777
RANJJVIMTOIWIN-UHFFFAOYSA-N
unii-f1klt23o3a, f1klt23o3a, chembl71917, 7-2,6-difluorophenyl methyl-4,7-dihydro-2-4-2-methyl-1-oxopropyl amino phenyl-3-methyl phenylmethyl amino methyl-4-oxo-thieno 2,3-b pyridine-5-carboxylic acid 1-methylethyl ester, d02nco, isopropyl 3-benzyl methyl amino methyl-7-2,6-difluorophenyl methyl-2-4-2-methylpropanoylamino phenyl-4-oxo-thieno 2,3-b pyridine-5-carboxylate, isopropyl 3-n-benzyl-n-methylaminomethyl-7-2,6-difluorobenzyl-4,7-dihydro-2-4-isobutyrylaminophenyl-4-oxothieno 2,3-b pyridine-5-carboxylate hydrochloride, propan-2-yl 3-benzyl methyl amino methyl-7-2,6-difluorophenyl methyl-2-4-2-methylpropanoylamino phenyl-4-oxothieno 2,3-b pyridine-5-carboxylate, thieno 2,3-b pyridine-5-carboxylic acid, 7-2,6-difluorophenyl methyl-4,7-dihydro-2-4-2-methyl-1-oxopropyl amino phenyl-3-methyl phenylmethyl amino methyl-4-oxo-, 1-methylethyl ester, hydrochloride, 3-benzyl-methyl-amino-methyl-7-2,6-difluoro-benzyl-2-4-isobutyrylamino-phenyl-4-oxo-4,7-dihydro-thieno 2,3-b pyridine-5-carboxylic acid isopropyl ester; hydrochloride
9874838
propan-2-yl 3-[[benzyl(methyl)amino]methyl]-7-[(2,6-difluorophenyl)methyl]-2-[4-(2-methylpropanoylamino)phenyl]-4-oxothieno[2,3-b]pyridine-5-carboxylate
CC(C)C(=O)NC1=CC=C(C=C1)C2=C(C3=C(S2)N(C=C(C3=O)C(=O)OC(C)C)CC4=C(C=CC=C4F)F)CN(C)CC5=CC=CC=C5

Description

GnRH receptor antagonist

Potent, orally active and non-peptide gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist (IC50 values are 0.2, 4.0 and 60 nM for human, monkey and rat GnRH receptors respectively). Inhibits LH release in vitro (IC50 = 100 nM) and reduces plasma LH concentration in castrated male cynomolgus monkeys.
Quantity 1 mg
Formula Weight 657.77
Percent Purity >98%
Chemical Name or Material T 98475

Safety and Handling

Recommended Storage Desiccate at +4°C
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